{"id":40,"date":"2016-10-26T11:01:44","date_gmt":"2016-10-26T11:01:44","guid":{"rendered":"http:\/\/eventi.uniurb.it\/esmec\/?page_id=40"},"modified":"2016-12-20T16:37:51","modified_gmt":"2016-12-20T16:37:51","slug":"programme-2016","status":"publish","type":"page","link":"https:\/\/eventi.uniurb.it\/esmec\/?page_id=40","title":{"rendered":"Programme"},"content":{"rendered":"<h3 class=\"p1\"><span class=\"s1\">SUNDAY, JUNE 26<\/span><\/h3>\n<p><strong>15.00 \u2013 18.30<\/strong><\/p>\n<p>Registration<\/p>\n<p><strong>19.00 \u2013 22.00<\/strong><\/p>\n<p>Poster Exhibition and Buffet Dinner<\/p>\n<h3 class=\"p1\"><span class=\"s1\">MONDAY, JUNE 27<\/span><\/h3>\n<p><strong>09.00 \u2013 09.20<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Opening of ESMEC 2016<\/span><\/p>\n<ul>\n<li class=\"p1\"><span class=\"s1\">Gabriele Costantino\u00a0\u2013 President of the Medicinal Chemistry Division of the Italian Chemical Society<\/span><\/li>\n<li class=\"p1\"><span class=\"s1\">Jordi Gracia\u2013\u00a0Member of the\u00a0EFMC Executive Committee<\/span><\/li>\n<li class=\"p1\"><span class=\"s1\">Carlo De Micheli\u00a0\u2013 Director of the European School of Medicinal Chemistry<\/span><\/li>\n<\/ul>\n<p class=\"p1\">Drug discovery: perspectives in the war on cancer<\/p>\n<ul>\n<li class=\"p1\"><span class=\"s1\">Marco Mor\u00a0\u2013 University of Parma &#8211;\u00a0Parma (I)<\/span><\/li>\n<li class=\"p1\"><span class=\"s1\">Antonio Macchiarulo\u00a0\u2013\u00a0University of Perugia &#8211;\u00a0Perugia\u00a0(I)<\/span><\/li>\n<\/ul>\n<p><strong>09.20 \u2013 09.30<\/strong><\/p>\n<p>Introduction to the session<\/p>\n<p><strong>09.30 \u2013 10.15<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Giulio Draetta\u00a0\u2013 University of Texas-\u00a0Houston (USA)<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\">Changing paradigms in cancer treatment \u2013 drug discovery challenges<\/span><\/p>\n<p class=\"p1\"><strong>10.15 \u2013 11.00<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Paul W. Manley\u00a0\u2013 Novartis Pharma &#8211;\u00a0Basel (CH)<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\">Discovery of Imatinib and Nilotinib: Targeted ABL kinase inhibitors for the treatment of leukemia<\/span><\/p>\n<p><strong>11.00 \u2013 11.30<\/strong><\/p>\n<p>Coffee Break<\/p>\n<p><strong>11.30 \u2013 12.15<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Gianluca Papeo\u00a0\u2013 Nerviano Medical Sciences &#8211;\u00a0Milan (I)<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\">Leveraging DNA Repair defects of Cancer Cells: the Case of PARP Inhibitors<\/span><\/p>\n<p class=\"p1\"><strong>12.15 \u2013 13.00<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Manlio Palumbo\u00a0\u2013 University of Padova &#8211;\u00a0Padova (I)<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\">Innovative drugs based on nucleic acids<\/span><\/p>\n<p class=\"p1\"><strong>13.00 \u2013 14.30<\/strong><\/p>\n<p class=\"p1\">Lunch<\/p>\n<p class=\"p1\"><strong>14.30 \u2013 16.00<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Gilberto Spadoni\u00a0\u2013 University of\u00a0Urbino \u2013 Urbino (I)<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\">Poster Session I<\/span><\/p>\n<p class=\"p1\"><strong>16.00 \u2013 18.30<\/strong><\/p>\n<p class=\"p1\">Case Study \u2013 Session I<\/p>\n<p class=\"p1\"><strong>20.30<\/strong><\/p>\n<p class=\"p1\">Dinner<\/p>\n<h3 class=\"p1\">TUESDAY, JUNE 28<\/h3>\n<p><strong>09.00 \u2013 09.15<\/strong><\/p>\n<p>Introduction to the Session<\/p>\n<p>Protein-protein interactions: structures and druggability<\/p>\n<ul>\n<li class=\"p1\"><span class=\"s1\">Maria Laura Bolognesi\u00a0\u2013 University of\u00a0Bologna &#8211;\u00a0Bologna (I)<\/span><\/li>\n<li class=\"p1\"><span class=\"s1\">Stefania Butini\u00a0\u2013 University of\u00a0Siena &#8211;\u00a0Siena (I)<\/span><\/li>\n<\/ul>\n<p><strong>09.15 \u2013 10.00<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Thomas L. Blundell\u2013 University of Cambridge \u2013 Cambridge\u00a0(UK)<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\">Protein-Protein Interactions: Structures and Druggability<\/span><\/p>\n<p class=\"p1\"><strong>10.00 \u2013 10.45<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Maurizio Pellecchia\u00a0\u2013 UCR School of Medicine \u2013 Riverside (USA)<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\">Protein-protein interactions: challenges and opportunities for the\u00a0 development of novel therapeutics<\/span><\/p>\n<p class=\"p1\"><strong>10.45 \u2013 11.15<\/strong><\/p>\n<p class=\"p1\">Coffee Break<\/p>\n<p class=\"p1\"><strong>11.15 \u2013 12.00<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Maurizio Pellecchia\u00a0\u2013 UCR School of Medicine \u2013 Riverside (USA)<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\">Modern drug discovery technologies to tackle protein-protein\u00a0 interactions<\/span><\/p>\n<p class=\"p1\"><strong>12.00 \u2013 12.45<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Francesca Bernardini\u00a0\u2013 Polyphor Ltd \u2013 Allschwil (CH)<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\">A Novel Class of Antibiotics against MDR Gram-negative ESKAPE Pathogens<\/span><\/p>\n<p class=\"p1\"><strong>12.45 \u2013 14.00<\/strong><\/p>\n<p class=\"p1\">Lunch<\/p>\n<p class=\"p1\"><strong>14.00 \u2013 15.30<\/strong><\/p>\n<p class=\"p1\">Poster Session II<\/p>\n<p class=\"p1\">Gilberto Spadoni\u00a0\u2013 University of\u00a0Urbino \u2013 Urbino (I<\/p>\n<p class=\"p1\"><strong>15.30 -18.30<\/strong><\/p>\n<p class=\"p1\">Case Study \u2013 Session II<\/p>\n<p class=\"p1\"><strong>20.30<\/strong><\/p>\n<p class=\"p1\">Dinner<\/p>\n<h3 class=\"p1\"><\/h3>\n<h3 class=\"p1\"><span class=\"s1\">WEDNESDAY, JUNE 29<\/span><\/h3>\n<p><strong>09.00 \u2013 09.15<\/strong><\/p>\n<p>Introduction to the Session<\/p>\n<p>New avenues in Carbohydrate Chemistry<\/p>\n<ul>\n<li class=\"p1\"><span class=\"s1\">Fabrizio Micheli\u00a0&#8211;\u00a0Aptuit S.r.l. &#8211;\u00a0Verona (I)<\/span><\/li>\n<li class=\"p1\"><span class=\"s1\">Giampiero Spalluto\u00a0\u2013 University of Trieste \u2013 Trieste\u00a0(I)<\/span><\/li>\n<\/ul>\n<p><strong>09.15 \u2013 10.00<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Sabine Flitsch\u00a0\u2013 University of Manchester-\u00a0Manchester\u00a0(UK)<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\">Enzymatic Synthesis of Glycoconjugates<\/span><\/p>\n<p class=\"p1\"><strong>10.00 \u2013 10.45<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Hermen Overkleeft\u00a0\u2013 University of Leiden-\u00a0Leiden (NL)<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\">Chemical biology and medicinal chemistry of glycosphingolipid metabolism<\/span><\/p>\n<p class=\"p1\"><strong>10.45 \u2013 11.15<\/strong><\/p>\n<p class=\"p1\">Coffee Break<\/p>\n<p class=\"p1\"><strong>11.15 \u2013 12.00<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Carlo Unverzagt\u00a0\u2013 University of Bayreuth &#8211;\u00a0Bayreth\u00a0(D)<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\">Convergent synthesis of glycoproteins \u2013 biologics from scratch<\/span><\/p>\n<p class=\"p1\"><strong>12.00 \u2013 12.45<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Laura Cipolla\u00a0\u2013 University of\u00a0Milan Bicocca\u00a0&#8211;\u00a0Milan (I)<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\">Glycochemistry and tissue regeneration: challenges and opportunities<\/span><\/p>\n<p class=\"p1\"><strong>12.45 \u2013 14.00<\/strong><\/p>\n<p class=\"p1\">Lunch<\/p>\n<p class=\"p1\"><strong>14.00 \u2013 15.00<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Mario Varasi\u00a0\u2013 Fondazione-Istituto FIRC di Oncologia Molecolare, Milan (I)\u00a0<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\">2015 approved drugs: To market! To market!<\/span><\/p>\n<p><strong>15.00 \u2013 18.00<\/strong><\/p>\n<p>Workshop<\/p>\n<p><strong>20.30<\/strong><\/p>\n<p>Dinner<\/p>\n<p>&nbsp;<\/p>\n<h3 class=\"p1\">THURSDAY, JUNE\u00a030<\/h3>\n<p><strong>09.00 \u2013 09.15<\/strong><\/p>\n<p>Introduction to the Session<\/p>\n<p>Hot Topics<\/p>\n<ul>\n<li class=\"p1\"><span class=\"s1\">Jordi Gracia\u00a0\u2013 Almirall, S.A. \u2013 Sant Feliu de Llobregat (E)<\/span><\/li>\n<li class=\"p1\"><span class=\"s1\">Gilberto Spadoni\u00a0\u2013 University of\u00a0Urbino \u2013 Urbino\u00a0(I)<\/span><\/li>\n<\/ul>\n<p><strong>09.15 \u2013 10.00<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Marie-Priscille Brun\u00a0\u2013 Sanofi \u2013 Vitry-sur Seine (F)<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\">Antibody Drug Conjugates: a new wave of anti-cancer drugs<\/span><\/p>\n<p class=\"p1\"><strong>10.00 \u2013 10.45<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Stefano Salmaso\u00a0\u2013 University of Padova &#8211;\u00a0Padova (I)<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\">Supramolecular responsive\u00a0 architectures for smart tumor targeting<\/span><\/p>\n<p class=\"p1\"><strong>10.45 \u2013 11.15<\/strong><\/p>\n<p class=\"p1\">Coffee Break<\/p>\n<p class=\"p1\"><strong>11.15 \u2013 12.00<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Yves P. Auberson\u00a0\u2013 Novartis \u2013 Basel (CH)<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\">Medicinal chemists don\u2019t just make drugs \u2013 the art of developing medical imaging agents.<\/span><\/p>\n<p class=\"p1\"><strong>12.00 \u2013 12.45<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Alleyn Plowright\u00a0&#8211;\u00a0AstraZeneca \u00a0&#8211; M\u00f6lndal (S)<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\">Discovery of Novel Molecules for Therapeutic Heart Regeneration<\/span><\/p>\n<p><strong>12.45 \u2013 14.00<\/strong><\/p>\n<p>Lunch<\/p>\n<p><strong>14.00 \u2013 18.00<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Mario Varasi\u00a0\u2013 Fondazione-Istituto FIRC di Oncologia Molecolare, Milan (I)<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\"><b>Presentation and Discussion of Selected Posters<\/b><\/span><\/p>\n<p class=\"p1\"><strong>18.00<\/strong><\/p>\n<p class=\"p1\"><span class=\"s1\">Carlo De Micheli &#8211; University of\u00a0Milan \u2013 Milan\u00a0(I) \u2013 ESMEC Director &#8211;<\/span><\/p>\n<p class=\"p1\"><span class=\"s1\"><b>Concluding Remarks<\/b><\/span><\/p>\n<p class=\"p1\"><strong>20.30<\/strong><\/p>\n<p class=\"p1\">Gala Dinner<\/p>\n<h3 class=\"p1\"><span class=\"s1\">FRIDAY, JULY 1<\/span><\/h3>\n<p>Leaving of participants<\/p>\n","protected":false},"excerpt":{"rendered":"<p>SUNDAY, JUNE 26 15.00 \u2013 18.30 Registration 19.00 \u2013 22.00 Poster Exhibition and Buffet Dinner MONDAY, JUNE 27 09.00 \u2013 09.20 Opening of ESMEC 2016 Gabriele Costantino\u00a0\u2013 President of the Medicinal Chemistry Division of the Italian Chemical Society Jordi Gracia\u2013\u00a0Member of the\u00a0EFMC Executive Committee Carlo De Micheli\u00a0\u2013 Director of the European School of Medicinal Chemistry [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"parent":67,"menu_order":10,"comment_status":"closed","ping_status":"closed","template":"","meta":{"_et_pb_use_builder":"","_et_pb_old_content":"","_et_gb_content_width":"","footnotes":""},"class_list":["post-40","page","type-page","status-publish","hentry"],"_links":{"self":[{"href":"https:\/\/eventi.uniurb.it\/esmec\/index.php?rest_route=\/wp\/v2\/pages\/40","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/eventi.uniurb.it\/esmec\/index.php?rest_route=\/wp\/v2\/pages"}],"about":[{"href":"https:\/\/eventi.uniurb.it\/esmec\/index.php?rest_route=\/wp\/v2\/types\/page"}],"author":[{"embeddable":true,"href":"https:\/\/eventi.uniurb.it\/esmec\/index.php?rest_route=\/wp\/v2\/users\/1"}],"replies":[{"embeddable":true,"href":"https:\/\/eventi.uniurb.it\/esmec\/index.php?rest_route=%2Fwp%2Fv2%2Fcomments&post=40"}],"version-history":[{"count":13,"href":"https:\/\/eventi.uniurb.it\/esmec\/index.php?rest_route=\/wp\/v2\/pages\/40\/revisions"}],"predecessor-version":[{"id":176,"href":"https:\/\/eventi.uniurb.it\/esmec\/index.php?rest_route=\/wp\/v2\/pages\/40\/revisions\/176"}],"up":[{"embeddable":true,"href":"https:\/\/eventi.uniurb.it\/esmec\/index.php?rest_route=\/wp\/v2\/pages\/67"}],"wp:attachment":[{"href":"https:\/\/eventi.uniurb.it\/esmec\/index.php?rest_route=%2Fwp%2Fv2%2Fmedia&parent=40"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}