{"id":1352,"date":"2023-11-10T08:49:19","date_gmt":"2023-11-10T08:49:19","guid":{"rendered":"https:\/\/eventi.uniurb.it\/esmec\/?page_id=1352"},"modified":"2024-07-02T06:55:56","modified_gmt":"2024-07-02T06:55:56","slug":"programme","status":"publish","type":"page","link":"https:\/\/eventi.uniurb.it\/esmec\/?page_id=1352","title":{"rendered":"Programme"},"content":{"rendered":"<p>[et_pb_section fb_built=&#8221;1&#8243; _builder_version=&#8221;4.14.2&#8243; _module_preset=&#8221;default&#8221; global_colors_info=&#8221;{}&#8221;][et_pb_row _builder_version=&#8221;4.14.2&#8243; _module_preset=&#8221;default&#8221; global_colors_info=&#8221;{}&#8221;][et_pb_column type=&#8221;4_4&#8243; _builder_version=&#8221;4.14.2&#8243; _module_preset=&#8221;default&#8221; global_colors_info=&#8221;{}&#8221;][et_pb_text _builder_version=&#8221;4.14.2&#8243; _module_preset=&#8221;default&#8221; global_colors_info=&#8221;{}&#8221;]<\/p>\n<div class=\"et_pb_column et_pb_column_1_2 et_pb_column_8  et_pb_css_mix_blend_mode_passthrough et-last-child\">\n<div class=\"et_pb_module et_pb_text et_pb_text_4  et_pb_text_align_left et_pb_bg_layout_light\">\n<div class=\"et_pb_text_inner\">\n<p>&nbsp;<\/p>\n<p><strong>SUNDAY, JUNE 30<\/strong><\/p>\n<p>15.00 \u2013 18.30 Registration<\/p>\n<p>19.00 \u2013 22.00 Putting up of Posters and Dinner<\/p>\n<p>&nbsp;<\/p>\n<p><strong>MONDAY, JULY 1<\/strong><\/p>\n<p>09.00 \u2013 09.20 Opening of ESMEC 2024<br \/>Giorgio CALCAGNINI \u2013 Rector of the University of Urbino Carlo Bo<br \/>Luc VAN HIJFTE \u2013 President of the European Federation for Medicinal Chemistry and Chemical Biology<br \/>Maria Laura BOLOGNESI \u2013 President of the Medicinal Chemistry Division of the Italian Chemical Society<br \/>Marco MACCHIA \u2013 Director of the European School of Medicinal Chemistry<\/p>\n<p>MAKE IT UNBREAKABLE! COVALENT APPROACH IN DRUG DISCOVERY<\/p>\n<p>Co-chair: Andrea CAVALLI \u2013 University of Bologna (I)<br \/>Gianluca PAPEO \u2013 Nerviano Medical Sciences (I)<\/p>\n<p>09.20 \u2013 09.30 Introduction to the Session<\/p>\n<p>09.30 \u2013 10.15 Alessio LODOLA \u2013 University of Parma (I)<br \/>Models for the discovery of covalent inhibitors<\/p>\n<p>10.15 \u2013 11.00 Chiara BORSARI \u2013 University of Milan (I)<br \/>Integration of medicinal chemistry and chemical biology in the development of covalent<br \/>chemical probes<\/p>\n<p>11.00 \u2013 11.30 Coffee Break<\/p>\n<p>11.30 \u2013 12.15 Annamaria MARTORANA \u2013 University of Palermo (I)<br \/>Targeting Sars-Cov-2 Main protease in the treatment of COVID-19: focus on covalent<br \/>inhibition<\/p>\n<p>12.15 \u2013 13.00 Francesco CASUSCELLI \u2013 Nerviano Medical Sciences, Milan (I)<br \/>Leveraging Covalent Approaches for the Discovery and Drug Development of Dual<br \/>IDH1\/2 Second Generation Inhibitors<\/p>\n<p>13.00 \u2013 15.00 Lunch<\/p>\n<p>15.00 \u2013 17.00 Workshop: PICK YOUR FAVORITE ELECTROPHILE! FROM REACTIVITY SCALE TO COVALENT ADDUCT STRUCTURES<br \/>Chiara BORSARI \u2013 University of Milan (I)<br \/>Alessio LODOLA \u2013 University of Parma (I)<\/p>\n<p>17.00 \u2013 18.00 Poster Session <br \/>Chairperson: Gilberto SPADONI \u2013 University of Urbino Carlo Bo (I)<\/p>\n<p>20.00 Dinner<\/p>\n<p>21.00 Walking tour of the historic center of Urbino, UNESCO heritage site\u2003<\/p>\n<p><strong>TUESDAY, JULY 2<\/strong><\/p>\n<p>CLICK-AND-TAG: HOW BIOORTHOGONAL CHEMISTRY IS TRANSFORMING DRUG DISCOVERY<\/p>\n<p>Co-chair: Stephanie FEDERICO \u2013 University of Trieste (I)<br \/>Antimo GIOIELLO \u2013 University of Perugia (I)<\/p>\n<p>09.00 \u2013 09.15 Introduction to the Session<\/p>\n<p>09.15 \u2013 10.00 Helen OSBORN \u2013 University of Reading (UK)<br \/>Designing chemical reactions for use in living systems: the role of bioorthogonal chemistry<\/p>\n<p>10.00 \u2013 10.45 Anja PALMANS \u2013 Eindhoven University of Technology (NL)<br \/>Bioorthogonal catalysis for medicinal chemistry applications<\/p>\n<p>10.45 \u2013 11.15 Coffee Break<\/p>\n<p>11.15 \u2013 12.00 Fr\u00e9d\u00e9ric TARAN \u2013 Paris-Saclay University (F)<br \/>In vivo chemistry for diagnostic and therapeutic applications<\/p>\n<p>12.00 \u2013 12.45 Milan VRABEL \u2013 Czech Academy of Sciences, Prague (CZ)<br \/>Developing new bioorthogonal reactions: Expanding the toolbox for biomedical research<\/p>\n<p>12.45 \u2013 14.30 Lunch<\/p>\n<p>14.30 \u2013 16.00 Workshop: HOW TO TRANSLATE MEDCHEM DISCOVERIES INTO INNOVATION<br \/>Elisabetta Zaccaro \u2013 Notarbartolo &amp; Gervasi, Milan (I)<br \/>Marco Borgogno \u2013 IAMA Therapeutics, Genoa (I)<\/p>\n<p>16.00 Assemblea della sezione Giovani della Divisione di Chimica Farmaceutica della SCI<\/p>\n<p>17.00 \u2013 18.00 Poster Session <br \/>Chairperson: Gilberto SPADONI \u2013 University of Urbino Carlo Bo (I)<\/p>\n<p>19.45 Dinner<\/p>\n<p>21.00 Guided tour of the Ducal Palace<\/p>\n<p>&nbsp;<\/p>\n<p><strong>WEDNESDAY, JULY 3<\/strong><\/p>\n<p>UNUSUAL ELEMENTS AND FUNCTIONAL GROUPS SHAPING THE FUTURE OF MEDICINAL CHEMISTRY<\/p>\n<p>Co-chair: Paolo GRIECO \u2013 University of Naples Federico II (I)<br \/>Tracey PIRALI \u2013 University of Piemonte Orientale (I)<\/p>\n<p>09.00 \u2013 09.15 Introduction to the Session<\/p>\n<p>09.15 \u2013 10.00 Gian Cesare TRON \u2013 University of Piemonte Orientale (I)<br \/>Lost and found: (Re)discovering the potential of neglected functional groups in medicinal chemistry. A focus on isocyanides<\/p>\n<p>10.00 \u2013 10.45 Jack ROWBOTHAM \u2013 University of Manchester (UK)<br \/>Meeting the challenges of heavy drug synthesis with biocatalytic asymmetric deuteration<\/p>\n<p>10.45 \u2013 11.15 Coffee Break<\/p>\n<p>11.15 \u2013 12.00 Evamarie HEY-HAWKINS \u2013 Leipzig University (D)<br \/>Carborane-containing drugs: New keys for old locks<\/p>\n<p>12.00 \u2013 12.45 Mauro ADAMO \u2013 University of Medicine and Health Science, Dublin (IE)<br \/>Introduction of fluorine on small and large molecules: Opportunities for drug discovery and lead development<\/p>\n<p>12.45 \u2013 14.30 Lunch<\/p>\n<p>14.30 \u2013 17.00 Round Table: The Future of Medicinal Chemistry: the opinion of emerging voices (Open Webinar)<\/p>\n<p>Chairperson: Maria Laura BOLOGNESI \u2013 President of the Medicinal Chemistry Division of the Italian Chemical Society<\/p>\n<p>Participants: Chiara BORSARI \u2013 Universit\u00e0 degli Studi di Milano (I)<br \/>Matthias GEHRINGER \u2013 Eberhard Karls Universit\u00e4t T\u00fcbingen (D)<br \/>Luca LARAIA \u2013 Technical University of Denmark (DE)<br \/>Sebastian OEHLER \u2013 Philochem AG (CH)<br \/>Andrea TESTA \u2013 Amphista Therapeutics Limited (UK)<\/p>\n<p>Beatriz DE PASCUAL-TERESA \u2013 University CEU San Pablo, Madrid (E)<\/p>\n<p>17.00 \u2013 17.30 Fourth Edition of the ESMEC Alumni Award (Open Webinar)<\/p>\n<p>Chairperson: Maria Laura BOLOGNESI \u2013 President of the Medicinal Chemistry Division of the Italian Chemical Society<\/p>\n<p>20.30 Social Dinner<\/p>\n<p>&nbsp;<\/p>\n<p><strong>THURSDAY, JULY 4<\/strong><\/p>\n<p>Chairperson: Beatriz DE PASCUAL-TERESA, University CEU San Pablo, Madrid (E)<\/p>\n<p>09.00 \u2013 10.00 Tiziano BANDIERA \u2013 Istituto Italiano di Tecnologia, Genoa (I)<br \/>Market watch: new drug approval in 2023 and synthetic strategies<\/p>\n<p>10.00 \u2013 10.30 Coffee Break<\/p>\n<p>10.30 \u2013 10.45 Michele MARI \u2013 University of Urbino Carlo Bo (I)<br \/>EFMC-YSN: join the young scientists network!<\/p>\n<p>10.45 \u2013 12.45 Chairperson: Gilberto SPADONI \u2013 University of Urbino Carlo Bo (I)<br \/>Selected oral lectures by participants:<br \/>Cosentino Giuseppe, University of Catania<br \/>Cursaro Ilaria, University of Siena<br \/>Giannessi Lisa, University of Parma<br \/>Lammers Rob F., Leiden University, NL<br \/>Madruga Enrique, University Computense Madrid<br \/>Masoni Samuele, University of Pisa<br \/>Persico Margherita, University of Trieste<\/p>\n<p><span style=\"font-size: 14px;\">12.45 \u2013 13.15 Marco MACCHIA \u2013 University of Pisa (I) \u2013 Director of ESMEC\u00a0<\/span><\/p>\n<p>Awards of selected posters<br \/>Concluding remarks<\/p>\n<p>13.15 Lunch and leaving<\/p>\n<\/div>\n<\/div>\n<\/div>\n<p>[\/et_pb_text][\/et_pb_column][\/et_pb_row][\/et_pb_section]<\/p>\n","protected":false},"excerpt":{"rendered":"<p>&nbsp; SUNDAY, JUNE 30 15.00 \u2013 18.30 Registration 19.00 \u2013 22.00 Putting up of Posters and Dinner &nbsp; MONDAY, JULY 1 09.00 \u2013 09.20 Opening of ESMEC 2024Giorgio CALCAGNINI \u2013 Rector of the University of Urbino Carlo BoLuc VAN HIJFTE \u2013 President of the European Federation for Medicinal Chemistry and Chemical BiologyMaria Laura BOLOGNESI \u2013 [&hellip;]<\/p>\n","protected":false},"author":3,"featured_media":0,"parent":1337,"menu_order":20,"comment_status":"closed","ping_status":"closed","template":"","meta":{"_et_pb_use_builder":"on","_et_pb_old_content":"","_et_gb_content_width":"","footnotes":""},"class_list":["post-1352","page","type-page","status-publish","hentry"],"_links":{"self":[{"href":"https:\/\/eventi.uniurb.it\/esmec\/index.php?rest_route=\/wp\/v2\/pages\/1352","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/eventi.uniurb.it\/esmec\/index.php?rest_route=\/wp\/v2\/pages"}],"about":[{"href":"https:\/\/eventi.uniurb.it\/esmec\/index.php?rest_route=\/wp\/v2\/types\/page"}],"author":[{"embeddable":true,"href":"https:\/\/eventi.uniurb.it\/esmec\/index.php?rest_route=\/wp\/v2\/users\/3"}],"replies":[{"embeddable":true,"href":"https:\/\/eventi.uniurb.it\/esmec\/index.php?rest_route=%2Fwp%2Fv2%2Fcomments&post=1352"}],"version-history":[{"count":9,"href":"https:\/\/eventi.uniurb.it\/esmec\/index.php?rest_route=\/wp\/v2\/pages\/1352\/revisions"}],"predecessor-version":[{"id":1466,"href":"https:\/\/eventi.uniurb.it\/esmec\/index.php?rest_route=\/wp\/v2\/pages\/1352\/revisions\/1466"}],"up":[{"embeddable":true,"href":"https:\/\/eventi.uniurb.it\/esmec\/index.php?rest_route=\/wp\/v2\/pages\/1337"}],"wp:attachment":[{"href":"https:\/\/eventi.uniurb.it\/esmec\/index.php?rest_route=%2Fwp%2Fv2%2Fmedia&parent=1352"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}